SCHEMBL7274265

SCHEMBL7274265

COc1c(C)cc(CC#N)c(-c2ccccc2)c1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 6/20 0.39
PDE4A P27815 5/20 0.39
PDE4C Q08493 5/20 0.39
PDE4D Q08499 5/20 0.39
HPGD P15428 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
LMNA P02545 1/20 0.34
MAT2A P31153 1/20 0.34
ALDH1A1 P00352 3/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
CYP3A4 P08684 1/20 0.33
SQOR Q9Y6N5 2/20 0.33
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ABCB1 P08183 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274626 0.81 PDE4B (0.47) PDE4BPDE4APDE4CPDE4DHPGD
SCHEMBL7274689 0.78 SMN1; SMN2 (0.42) PDE4BPDE4APDE4CPDE4DHPGD
SCHEMBL11300639 0.76 ALDH1A1 (0.31) ALDH1A1
SCHEMBL27748134 0.73 IMPDH2 (0.33) ALDH1A1
SCHEMBL9080677 0.68 ALDH1A1 (0.40) HPGDKDM4EGAAALDH1A1TSHR
SCHEMBL29788016 0.68 FFAR2 (0.48) PDE4BPDE4APDE4CPDE4DKDM4E
SCHEMBL29473773 0.67 PDE4B (0.48) PDE4BPDE4APDE4CPDE4DHPGD
SCHEMBL411675 0.66 CNR1 (0.49) PDE4BPDE4APDE4CPDE4DHPGD
SCHEMBL31134292 0.66 PDE4B (0.47) PDE4BPDE4APDE4CPDE4DHPGD
SCHEMBL9376230 0.66 PDE4B (0.47) PDE4BPDE4APDE4CPDE4DHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed