SCHEMBL7274477

SCHEMBL7274477

O=C1OCc2nc3cc(Cl)ccc3c(O)c21

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 10/20 0.43
BCHE P06276 9/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CHRM1 P11229 1/20 0.43
EPHX2 P34913 1/20 0.43
C1R P00736 1/20 0.38
APEX1 P27695 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283362 0.89 L3MBTL1 (0.45) ACHEBCHEMEN1KMT2A
SCHEMBL29249103 0.81 ESR1 (0.52) ACHEMEN1KMT2A
SCHEMBL7274459 0.81 KMT2A (0.41) ACHEBCHEMEN1KMT2ACHRM1
SCHEMBL5014974 0.74 PDE1A (0.52) ACHEBCHEMEN1KMT2A
SCHEMBL29249095 0.69 MEN1 (0.51) MEN1KMT2A
SCHEMBL29249036 0.69 MEN1 (0.48) MEN1KMT2A
SCHEMBL29249055 0.65 MEN1 (0.52) ACHEMEN1KMT2AC1R
SCHEMBL7283059 0.65 KDM4E (0.46) ACHEMEN1KMT2A
SCHEMBL8133213 0.64 PDE3B (0.50) ACHEMEN1KMT2A
SCHEMBL9876043 0.64 ACHE (0.63) ACHEBCHEKMT2ACHRM1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481429-B1 Quinoline derivatives SS PHARMACEUTICAL CO (JP) 2001-01-24 EP disclosed
EP-0987262-A1 Quinoline derivatives SS PHARMACEUTICAL CO., LTD. (JP) 2000-03-22 EP disclosed
US-5300517-A Treating Alzheimer's SS PHARMACEUTICAL CO., LTD. (JP) 1994-04-05 US disclosed
US-5240934-A Cognition activators SS PHARMACEUTICAL CO., LTD. (JP) 1993-08-31 US disclosed
EP-0481429-A2 Quinoline derivatives SS PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed