SCHEMBL7274758

SCHEMBL7274758

CON(C)C(=O)C[C@H](NC(=O)OCc1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.49
TSHR P16473 4/20 0.49
ATM Q13315 2/20 0.49
ALDH1A1 P00352 3/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP1A2 P05177 2/20 0.48
POLB P06746 1/20 0.48
CYP2D6 P10635 1/20 0.48
CTSL P07711 2/20 0.48
CTSS P25774 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.47
CASP1 P29466 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CTSB P07858 1/20 0.46
CTSK P43235 1/20 0.46
OPRK1 P41145 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22982779 1.00 CYP3A4 (0.49) CYP3A4TSHRATMALDH1A1CYP2C9
SCHEMBL20993378 0.87 KMT2A (0.47) CYP3A4TSHRALDH1A1CYP2C9CYP2C19
SCHEMBL2342652 0.84 CTSK (0.51) ATMALDH1A1CTSLCTSSCASP1
SCHEMBL3414548 0.84 CTSK (0.51) ATMALDH1A1CTSLCTSSCASP1
SCHEMBL8382243 0.83 FAAH (0.46) ALDH1A1CYP2C19CYP1A2POLBKMT2A
SCHEMBL6958944 0.83 ATM (0.54) CYP3A4TSHRATMALDH1A1CYP2C9
SCHEMBL16201457 0.83 ATM (0.54) CYP3A4TSHRATMALDH1A1CYP2C9
SCHEMBL4125738 0.83 KMT2A (0.48) TSHRALDH1A1MEN1KMT2A
SCHEMBL7285800 0.82 ATM (0.55) CYP3A4TSHRATMALDH1A1CYP2C9
SCHEMBL6156731 0.82 CASP1 (0.60) ATMALDH1A1CYP1A2CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0361341-A2 Therapeutics for aids based on inhibitors of HIV protease MILES INC. (US) 1990-04-04 EP disclosed