SCHEMBL7276038

SCHEMBL7276038

CN1CCCCC1COC(=O)c1cn(C)c2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.58
CHRNA5 P30532 2/20 0.58
CHRNA7 P36544 2/20 0.58
CHRNA4 P43681 2/20 0.58
CYP1A2 P05177 1/20 0.55
CYP2C9 P11712 1/20 0.55
ALOX15 P16050 1/20 0.55
NFKB1 P19838 1/20 0.55
PMP22 Q01453 1/20 0.55
HTR4 Q13639 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
CNR1 P21554 1/20 0.53
CNR2 P34972 1/20 0.53
NR4A2 P43354 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
RAB9A P51151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16887920 0.86 NR4A2 (0.52) CHRNB2CHRNA5CHRNA7CHRNA4CYP1A2
SCHEMBL7276531 0.85 CNR1 (0.56) CHRNB2CHRNA5CHRNA7CHRNA4NPSR1
SCHEMBL7271018 0.85 CNR1 (0.57) CHRNB2CHRNA5CHRNA7CHRNA4CNR1
SCHEMBL7300604 0.80 HTR4 (0.69) CYP1A2CYP2C9ALOX15NFKB1PMP22
SCHEMBL7269469 0.79 CYP2D6 (0.60) CHRNB2CHRNA5CHRNA7CHRNA4CYP1A2
SCHEMBL8802608 0.79 CHRNB2 (0.57) CHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL7269463 0.79 CYP2D6 (0.60) CHRNB2CHRNA5CHRNA7CHRNA4CYP1A2
SCHEMBL7271039 0.79 CYP2D6 (0.60) CHRNB2CHRNA5CHRNA7CHRNA4CYP1A2
SCHEMBL9344429 0.78 HTR4 (0.67) CYP1A2CYP2C9ALOX15NFKB1PMP22
SCHEMBL7277894 0.78 CYP2D6 (0.62) CHRNB2CHRNA5CHRNA7CHRNA4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429984-B1 Indole derivatives NISSHIN FLOUR MILLING CO (JP) 1997-07-23 EP disclosed
US-5124324-A Psychological disorders, 5-hydroxy tryptamine antagonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-06-23 US disclosed
EP-0429984-A2 Indole derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-06-05 EP disclosed