SCHEMBL7277494

SCHEMBL7277494

COc1ccc2c(c1)CC(N)(C(=O)O)C2

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CXCR5 P32302 2/20 0.47
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HTR5A P47898 2/20 0.41
METAP1 P53582 1/20 0.41
POLA1 P09884 2/20 0.40
HSD17B10 Q99714 1/20 0.40
CA2 P00918 1/20 0.40
MAOB P27338 1/20 0.40
KDM4E B2RXH2 2/20 0.40
NOTUM Q6P988 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8345353 0.88 ADRA2A (0.47) CXCR5NPC1RAB9AHTR5APOLA1
SCHEMBL16836163 0.82 CXCR5 (0.51) CXCR5NPC1RAB9AMETAP1POLA1
SCHEMBL29346208 0.81 CXCR5 (0.33) CXCR5HSD17B10KDM4EALDH1A1MAPK1
SCHEMBL3309532 0.81 ALDH1A1 (0.41) CXCR5NPC1RAB9AHTR5AHSD17B10
SCHEMBL26402689 0.79 ADRA2A (0.40) CXCR5RAB9AHTR5APOLA1HSD17B10
Hydrochloric Acid SCHEMBL31435767 0.79 ADRA2A (0.40) CXCR5RAB9AHTR5APOLA1HSD17B10
Hydrochloric Acid SCHEMBL26127895 0.79 ADRA2A (0.40) CXCR5RAB9AHTR5APOLA1HSD17B10
SCHEMBL3307587 0.78 SMN1; SMN2 (0.52) CXCR5NPC1RAB9AHTR5AHSD17B10
SCHEMBL7277003 0.78 HSD17B1 (0.42) MAOBKDM4EALDH1A1CYP3A4
SCHEMBL23811628 0.78 DRD2 (0.45) HTR5AMETAP1POLA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766110-A INHIBITS ANGIOTENSIN CONVERTING ENZYME, HYPOTENSIVE AGENTS RYAN JAMES W (US) 1988-08-23 US disclosed
EP-0073143-B1 NOVEL COMPLEX AMIDO AND IMIDO DERIVATIVES OF CARBOXYALKYL PEPTIDES AND THIOETHERS AND ETHERS OF PEPTIDES Ryan, James Walter (US) 1985-11-21 EP disclosed
EP-0073143-A2 Novel complex amido and imido derivatives of carboxyalkyl peptides and thioethers and ethers of peptides Ryan, James Walter (US) 1983-03-02 EP disclosed
EP-0048159-A2 Novel carboxyalkyl peptides and thioethers and ethers of peptides as antihypertensive agents UNIVERSITY OF MIAMI (US) 1982-03-24 EP disclosed