SCHEMBL7277767

SCHEMBL7277767

O=C(N[C@@H](Cc1ccccc1)[C@@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)c1ccccn1)c1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.55
HTT P42858 3/20 0.50
KDM4E B2RXH2 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CA2 P00918 1/20 0.50
MAPT P10636 1/20 0.50
CTSD P07339 3/20 0.48
EPHX2 P34913 1/20 0.48
KMT2A Q03164 1/20 0.48
USP30 Q70CQ3 1/20 0.47
LMNA P02545 1/20 0.46
OPRK1 P41145 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8853761 0.87 CA2 (0.66) CA2CTSD
SCHEMBL6447454 0.87 CA2 (0.66) CA2CTSD
SCHEMBL29648527 0.87 CA2 (0.66) CA2CTSD
SCHEMBL5805400 0.83 PYGL (0.57) PSMB5HTTKDM4ESMN1; SMN2CA2
SCHEMBL21623659 0.81 PSMB5 (0.62) PSMB5HTTKDM4ESMN1; SMN2CA2
SCHEMBL9554481 0.81 PSMB5 (0.62) PSMB5HTTKDM4ESMN1; SMN2CA2
SCHEMBL24862890 0.79 CAPN1 (0.56) PSMB5HTTKDM4ESMN1; SMN2MAPT
SCHEMBL6931878 0.79 CTRB1 (0.59) PSMB5
SCHEMBL6448868 0.78 ROCK2 (0.56) HTTKDM4EMAPTEPHX2TDP1
SCHEMBL8013304 0.78 PSMB5 (0.59) PSMB5USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed