SCHEMBL7280301

SCHEMBL7280301

CC(=O)N1CCC(N(C)Cc2ccccc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.63
JAK2 O60674 1/20 0.53
JAK1 P23458 1/20 0.53
AGTR2 P50052 2/20 0.52
RORC P51449 3/20 0.50
OPRM1 P35372 2/20 0.50
SIGMAR1 Q99720 1/20 0.50
NPY5R Q15761 1/20 0.49
KMT2A Q03164 2/20 0.48
GRIN2B Q13224 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MCHR1 Q99705 1/20 0.47
MEN1 O00255 1/20 0.46
UBE2M P61081 1/20 0.46
DCUN1D1 Q96GG9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26618018 0.92 KMT2A (0.55) LTA4HJAK2JAK1AGTR2RORC
SCHEMBL785972 0.90 JAK2 (0.54) LTA4HJAK2JAK1AGTR2OPRM1
SCHEMBL9451691 0.86 LTA4H (0.57) LTA4HRORCOPRM1KDM4E
Hydrochloric Acid SCHEMBL7468874 0.85 CHIA (0.50) LTA4HAGTR2OPRM1SIGMAR1NPY5R
SCHEMBL18424508 0.84 KMT2A (0.56) LTA4HJAK2JAK1AGTR2OPRM1
SCHEMBL14144125 0.83 JAK2 (0.52) LTA4HJAK2JAK1AGTR2OPRM1
SCHEMBL803527 0.81 JAK2 (0.74) JAK2JAK1KMT2AKDM4EMEN1
SCHEMBL20160113 0.81 ALDH1A1 (0.56) LTA4HJAK2JAK1AGTR2OPRM1
SCHEMBL16757240 0.81 KMT2A (0.69) RORCOPRM1KMT2AKDM4EALDH1A1
SCHEMBL7292853 0.80 L3MBTL3 (0.55) LTA4HJAK2JAK1AGTR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0457686-B1 Novel aminopiperidine, aminopyrrolidine and aminoperhydroazepine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1994-08-03 EP disclosed
US-5214055-A Analgesics, psychological disorders, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-05-25 US disclosed
US-5189045-A Antiserotonine agent ADIR ET COMPAGNIE (FR) 1993-02-23 US disclosed
EP-0457686-A1 Novel aminopiperidine, aminopyrrolidine and aminoperhydroazepine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-11-21 EP disclosed