SCHEMBL7280877

SCHEMBL7280877

CC1(Cl)Oc2c(C(=O)O)cc(Cl)cc2N(CCCc2ccccc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
ALDH2 P05091 2/20 0.40
ALDH3A1 P30838 2/20 0.40
PKM P14618 1/20 0.40
ADRA1D P25100 1/20 0.39
SLC5A2 P31639 1/20 0.39
TP53 P04637 3/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ELANE P08246 1/20 0.37
CTSG P08311 1/20 0.37
PRTN3 P24158 1/20 0.37
PARK7 Q99497 2/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
TGM2 P21980 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288574 0.94 ALDH1A1 (0.44) ALDH1A1ALDH2ALDH3A1ADRA1DSLC5A2
SCHEMBL7287349 0.80 MAPT (0.41) ALDH1A1SLC5A2TP53SMN1; SMN2ELANE
SCHEMBL7288496 0.79 GRM2 (0.40) SLC5A2ELANECTSGPRTN3PTGDR2
SCHEMBL7288613 0.78 ALDH1A1 (0.41) ALDH1A1ALDH2ALDH3A1PKMADRA1D
SCHEMBL7281540 0.78 NLRP3 (0.41) ALDH1A1TP53SMN1; SMN2CA2CA9
SCHEMBL7291581 0.78 SCN9A (0.43) ALDH1A1PKMTP53GSK3AGSK3B
Hydrochloric Acid SCHEMBL7280882 0.78 ALDH1A1 (0.40) ALDH1A1ALDH2ALDH3A1PKMADRA1D
SCHEMBL10427989 0.76 CA12 (0.39) SMN1; SMN2PTGDR2CA2CA9
Hydrochloric Acid SCHEMBL7290990 0.75 ELANE (0.43) ALDH1A1ALDH2ALDH3A1SLC5A2TP53
SCHEMBL9488302 0.74 DRD2 (0.40) ALDH1A1ALDH2ALDH3A1ADRA1DSLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0313393-B1 Benzoxazine compounds and pharmaceutical use thereof YOSHITOMI PHARMACEUTICAL (JP) 1994-03-16 EP disclosed
US-4892872-A ANTIEMETICS, ANTINAUSEA YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-01-09 US disclosed