SCHEMBL7280890

SCHEMBL7280890

COC(=O)CCc1ccc(-n2ncn(-c3ccc(C(=N)NC(=O)OC)cc3)c2=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 2/20 0.36
TSHR P16473 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
CYP11B1 P15538 5/20 0.33
CYP11B2 P19099 5/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
HSD17B3 P37058 1/20 0.32
PTPN1 P18031 3/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273458 0.88 ITGB3 (0.44) RPS6KA3
Hydrochloric Acid SCHEMBL7281884 0.87 ITGB3 (0.43) RPS6KA3
Hydrochloric Acid SCHEMBL8573867 0.87 ITGB3 (0.43) RPS6KA3
SCHEMBL7282163 0.85 PTPN1 (0.37) RPS6KA3HRH3ADRB2ADRB1PTPN1
SCHEMBL7281314 0.83 RPS6KA3 (0.39) RPS6KA3TSHRHRH3CYP11B1CYP11B2
SCHEMBL7273332 0.80 CYP11B2 (0.51) RPS6KA3TSHRHRH3CYP11B1CYP11B2
SCHEMBL7282680 0.80 CYP11B2 (0.51) RPS6KA3TSHRHRH3CYP11B1CYP11B2
SCHEMBL7274885 0.80 LMNA (0.35) RPS6KA3HRH3ADRB2ADRB1PTPN1
SCHEMBL7280894 0.79 F2 (0.43)
SCHEMBL7281654 0.78 KMT2A (0.40) HRH3ADRB2ADRB1HPGDPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed