SCHEMBL7282120

SCHEMBL7282120

CCc1nn(C)c2c1C(c1cccc(OC)c1OC)C(C(=O)OC)=C(C)N2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 5/20 0.50
GAA P10253 3/20 0.50
GLA P06280 1/20 0.50
PKM P14618 1/20 0.44
HSD17B10 Q99714 7/20 0.44
HPGD P15428 3/20 0.44
CASP1 P29466 2/20 0.44
CASP7 P55210 1/20 0.44
BAP1 Q92560 1/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
TSHR P16473 5/20 0.42
CYP2C9 P11712 4/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2C19 P33261 3/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 3/20 0.40
CYP1A2 P05177 2/20 0.40
HIF1A Q16665 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278442 0.93 ALDH1A1 (0.48) ALDH1A1KDM4EGAAGLAPKM
SCHEMBL7272107 0.88 GAA (0.48) ALDH1A1KDM4EGAAGLAPKM
SCHEMBL7272453 0.85 GAA (0.45) ALDH1A1KDM4EGAAGLAPKM
SCHEMBL7272727 0.84 ADORA3 (0.42) ALDH1A1KDM4EGAAHSD17B10HPGD
SCHEMBL7278457 0.77 ADORA3 (0.41) ALDH1A1KDM4EGAAHSD17B10HPGD
SCHEMBL7272955 0.76 ALDH1A1 (0.43) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL7280395 0.76 CACNA1F (0.56) ALDH1A1KDM4EGAAPKMHPGD
SCHEMBL7437834 0.75 GAA (0.46) ALDH1A1KDM4EGAAHSD17B10HPGD
SCHEMBL7273188 0.74 LMNA (0.52) ALDH1A1KDM4EGAAHSD17B10HPGD
SCHEMBL10367692 0.74 NR1I2 (0.56) ALDH1A1KDM4EGAAGLAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0114273-B1 NEW PHARMACOLOGICALLY ACTIVE PYRAZOLOPYRIDINES GRUPPO LEPETIT S.p.A. (IT) 1991-11-06 EP disclosed
US-4954508-A HYPOTENSIVE GRUPPO LEPETIT S.P.A. (IT) 1990-09-04 US disclosed