SCHEMBL7284247

SCHEMBL7284247

N#Cc1ccc(-c2ccc(OC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CCCc3ccccc3)nn2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.37
DRD4 P21917 1/20 0.37
HTR2A P28223 1/20 0.37
HRH1 P35367 1/20 0.37
OPRM1 P35372 1/20 0.37
FAAH O00519 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 2/20 0.34
ABCB1 P08183 1/20 0.34
HPGD P15428 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NR3C2 P08235 1/20 0.34
BCHE P06276 2/20 0.34
ACHE P22303 2/20 0.34
EP300 Q09472 2/20 0.34
DGAT1 O75907 1/20 0.33
ADORA2A P29274 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7276144 0.92 EP300 (0.37) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7285879 0.88 BCHE (0.33) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7338546 0.87 ITGB3 (0.39) OPRM1ALDH1A1TSHRSMN1; SMN2KCNH2
SCHEMBL7275504 0.86 ABCB1 (0.45) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7276469 0.86 ABCB1 (0.45) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7276043 0.85 EP300 (0.39) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7273402 0.84 ABCB1 (0.44) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7273518 0.81 ABCB1 (0.46) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7274473 0.81 HTR1A (0.37) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7280953 0.81 HRH3 (0.40) HTR1ADRD4HTR2AHRH1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed