SCHEMBL7284387

SCHEMBL7284387

COC(=O)C[C@@H]1C[C@@H](CNC(=O)c2cc(-c3ccc(C#N)cc3)n[nH]c2=O)N(CCCc2ccccc2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.34
DRD4 P21917 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
OPRM1 P35372 1/20 0.34
USP30 Q70CQ3 1/20 0.34
TACR3 P29371 1/20 0.34
CHRM4 P08173 1/20 0.34
TP53 P04637 1/20 0.33
DRD2 P14416 3/20 0.33
ABCB1 P08183 1/20 0.33
HPGD P15428 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
DRD3 P35462 3/20 0.33
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7277118 0.88 F2 (0.37) TP53DRD2
SCHEMBL7274708 0.85 CHRM4 (0.42) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7281347 0.83 DRD2 (0.35) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7278834 0.83 HTR1A (0.39) HTR1ACHRM4ABCB1HPGDABCG2
SCHEMBL7275850 0.81 ITGB3 (0.39)
SCHEMBL7275885 0.81 EP300 (0.40) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7284718 0.80 HTR1A (0.42) HTR1ADRD4DRD2DRD3
SCHEMBL7273748 0.80 HTR1A (0.38) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7273369 0.80 MAOA (0.38) HTR1ACHRM4DRD2DRD3MAPT
SCHEMBL7273026 0.80 NAMPT (0.40) HTR1ADRD4OPRM1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed