SCHEMBL7285181

SCHEMBL7285181

O=C(O)C[C@@H]1C[C@@H](CN2C(=O)c3ccccc3C2=O)N(CCCc2ccccc2)C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 2/20 0.41
TSHR P16473 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP1B1 Q16678 2/20 0.40
ALDH2 P05091 1/20 0.40
PKM P14618 1/20 0.40
ALDH3A1 P30838 1/20 0.40
MAPK1 P28482 1/20 0.40
CASP3 P42574 1/20 0.40
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
ASAH1 Q13510 1/20 0.38
ITGB3 P05106 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273909 0.84 TDP1 (0.44) TDP1L3MBTL1ALDH1A1TSHRSMN1; SMN2
SCHEMBL7282531 0.83 ALDH1A1 (0.45) ALDH1A1TSHRSMN1; SMN2MAPK1OPRD1
SCHEMBL7282112 0.82 TDP1 (0.43) TDP1L3MBTL1ALDH1A1TSHRCYP1B1
SCHEMBL7273681 0.82 ALDH1A1 (0.44) ALDH1A1TSHRSMN1; SMN2MAPK1OPRD1
SCHEMBL7275206 0.81 ALDH1A1 (0.43) ALDH1A1TSHRSMN1; SMN2MAPK1ADRA1A
SCHEMBL7282793 0.80 ALDH1A1 (0.45) ALDH1A1TSHRSMN1; SMN2MAPK1ADRA1A
SCHEMBL7273778 0.79 TBXA2R (0.39) ALDH1A1SMN1; SMN2PKM
SCHEMBL7281899 0.77 CASP3 (0.43) TDP1L3MBTL1ALDH1A1SMN1; SMN2CYP1B1
SCHEMBL7273271 0.77 ALDH1A1 (0.40) ALDH1A1TSHRSMN1; SMN2MAPK1ITGB3
SCHEMBL7274386 0.75 TDP1 (0.46) TDP1L3MBTL1ALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed