SCHEMBL7285654

SCHEMBL7285654

COc1ccc(-c2ccc(C#N)cc2)cc1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.54
CYP17A1 P05093 1/20 0.51
ACLY P53396 1/20 0.49
NAAA Q02083 2/20 0.47
PDGFRB P09619 1/20 0.47
PDGFRA P16234 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
KDM1A O60341 2/20 0.46
PI4KB Q9UBF8 1/20 0.46
TDP2 O95551 1/20 0.46
ERN1 O75460 1/20 0.46
FFAR1 O14842 1/20 0.45
ALPL P05186 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9061902 1.00 KIF11 (0.54) KIF11CYP17A1ACLYNAAAPDGFRB
SCHEMBL31128553 0.85 AR (0.51) KDM1AALDH1A1RAB9AAR
SCHEMBL313099 0.85 AR (0.51) KDM1AALDH1A1RAB9AAR
SCHEMBL9464193 0.83 CYP17A1 (0.61) CYP17A1PDGFRBPDGFRAKDM1ATDP2
SCHEMBL13802320 0.81 AR (0.50) KIF11ACLYPDGFRBPDGFRAKDM1A
SCHEMBL16945932 0.81 PTGS2 (0.47) KIF11ACLYPDGFRBPDGFRAKDM1A
SCHEMBL15420520 0.81 ALDH1A1 (0.47) PDGFRBPDGFRAKDM1API4KBMEN1
SCHEMBL15605813 0.80 CYP17A1 (0.58) CYP17A1NAAAPDGFRBPDGFRATDP2
SCHEMBL8883091 0.79 ACLY (0.49) KIF11ACLYKDM1AALPLALDH1A1
SCHEMBL7283993 0.79 KIF11 (0.58) KIF11ACLYAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed