SCHEMBL7288986

SCHEMBL7288986

Cc1ccc(N2CCN(CCCNc3ccc(Cl)cc3S)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
DRD2 P14416 7/20 0.46
MAPT P10636 2/20 0.45
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
TP53 P04637 1/20 0.44
CACNA1G O43497 1/20 0.43
DRD3 P35462 1/20 0.43
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7290150 0.88 CACNA1G (0.55) DRD2MAPTTP53CACNA1GDRD3
SCHEMBL2486143 0.79 HRH3 (0.70)
SCHEMBL7283381 0.78 CACNA1G (0.60) DRD2MAPTSLC6A4CACNA1GDRD3
SCHEMBL6843584 0.75 DRD2 (0.54) DRD4DRD2MAPTSLC6A2SLC6A4
SCHEMBL7283745 0.74 DRD3 (0.50) DRD4DRD2SLC6A2SLC6A4DRD3
SCHEMBL2512341 0.73 ACP1 (0.55) DRD2SLC6A2SLC6A4
SCHEMBL2488597 0.71 HRH3 (0.76)
SCHEMBL6846732 0.71 MAPT (0.54) DRD4KDM4EDRD2MAPTTP53
SCHEMBL11447942 0.70 HTR7 (0.60) DRD4DRD2MAPTSLC6A4TP53
SCHEMBL10995656 0.70 MAPT (0.58) KDM4EGAADRD2MAPTDRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609031-B1 Process for preparing benzothiazepine derivatives SHIONOGI & CO (JP) 1997-08-13 EP disclosed
EP-0609031-A1 Process for preparing benzothiazepine derivatives SHIONOGI & CO., LTD. (JP) 1994-08-03 EP disclosed