SCHEMBL7289944

SCHEMBL7289944

Cc1cc(C)c(C(Cl)C(N)=O)c(C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
F2 P00734 3/20 0.37
PRSS1 P07477 3/20 0.37
PRSS2 P07478 3/20 0.37
PRSS3 P35030 3/20 0.37
LMNA P02545 4/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
GAA P10253 1/20 0.34
ALOX5 P09917 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HTT P42858 1/20 0.33
TSHR P16473 1/20 0.33
POLB P06746 1/20 0.32
TPMT P51580 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27841663 0.81 ALDH1A1 (0.35) KDM4ELMNAALDH1A1MAPTGAA
SCHEMBL6807941 0.80 KDM4E (0.42) KDM4EF2PRSS1PRSS2PRSS3
SCHEMBL7279957 0.80 SMN1; SMN2 (0.31) SMN1; SMN2POLB
SCHEMBL1922886 0.79 HSP90AA1 (0.37) KDM4ELMNAALDH1A1TSHRPOLB
SCHEMBL7432717 0.77 ALDH1A1 (0.38) ALDH1A1MAPTGAAPOLB
SCHEMBL28303367 0.77 TPMT (0.38) KDM4EF2PRSS1PRSS2PRSS3
SCHEMBL28809532 0.77 KDM4E (0.39) KDM4EF2PRSS1PRSS2PRSS3
SCHEMBL30819282 0.72 LMNA (0.37) KDM4EF2PRSS1PRSS2PRSS3
SCHEMBL21259500 0.70 SLC6A2 (0.38) KDM4EF2PRSS1PRSS2PRSS3
SCHEMBL22298450 0.70 SLC6A2 (0.38) KDM4EF2PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed