SCHEMBL7290699

SCHEMBL7290699

COc1cc(C(=O)c2ccnc(Br)c2)c(C(OC)OC)cc1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.42
SENP6 Q9GZR1 4/20 0.42
SENP8 Q96LD8 3/20 0.42
SENP7 Q9BQF6 3/20 0.42
APAF1 O14727 2/20 0.42
NSD2 O96028 2/20 0.42
TDP2 O95551 1/20 0.42
PPP1CA P62136 1/20 0.42
SAE1 Q9UBE0 1/20 0.42
UBA2 Q9UBT2 1/20 0.42
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP1A2 P05177 4/20 0.38
CYP2C19 P33261 4/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 3/20 0.38
TSHR P16473 1/20 0.38
SRC P12931 3/20 0.37
TGFBR1 P36897 3/20 0.37
LCK P06239 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297929 0.85 RORB (0.39) CASP3SENP6SENP8SENP7APAF1
SCHEMBL7289967 0.82 LCK (0.50) CASP3SENP6SENP8SENP7APAF1
SCHEMBL7381304 0.79 LCK (0.41) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL7295979 0.79 PRKDC (0.44) CASP3SENP6SENP8SENP7APAF1
SCHEMBL7380165 0.74 TUBB1 (0.49) LMNA
SCHEMBL16773953 0.73 ACHE (0.40) CASP3SENP6SENP8SENP7APAF1
SCHEMBL28786825 0.71 LMNA (0.47) ALDH1A1L3MBTL1LMNAMAPT
SCHEMBL29584593 0.67 KDM4E (0.60) ALDH1A1L3MBTL1TSHRHPGDMAPT
SCHEMBL46685 0.67 KDM4E (0.60) ALDH1A1L3MBTL1TSHRHPGDMAPT
SCHEMBL16691026 0.67 ACHE (0.35) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848000-B1 Pharmaceutical pyridine derivatives, processes for preparing the same and intermediates therefor TANABE SEIYAKU CO (JP) 2002-06-12 EP disclosed
US-5965730-A SELECTIVE PHOSPHODIESTEARASE IV INHIBITOR HAVING BRONCHODIALATION AND ANTI-INFLAMMATORY ACTIVITY; PROPHYLAXIS AND TREATMENT OF ASTHMA TANABE SEIYAKU CO., LTD. (JP) 1999-10-12 US disclosed
EP-0848000-A1 Pharmaceutical pyridine derivatives, processes for preparing the same and intermediates therefor TANABE SEIYAKU CO., LTD. (JP) 1998-06-17 EP disclosed