SCHEMBL7294757

SCHEMBL7294757

Nc1ccc(Cc2cccs2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.52
ALDH1A1 P00352 1/20 0.52
TSHR P16473 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
TAAR1 Q96RJ0 1/20 0.52
CYP17A1 P05093 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
GFER P55789 1/20 0.41
ADRA1D P25100 2/20 0.41
LMNA P02545 1/20 0.41
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29337530 0.83 LTA4H (0.57) TAAR1CYP17A1CYP11B1CYP11B2ADRA2A
SCHEMBL45228 0.80 LMNA (0.50) ALDH1A1TSHRTDP1TAAR1ADRA1D
SCHEMBL10525378 0.79 L3MBTL1 (0.55) TAAR1ADRA2AADRA2BADRA2CADRA1D
SCHEMBL3238290 0.79 LMNA (0.62) ALDH1A1TAAR1ADRA1DLMNAPTGS1
SCHEMBL923302 0.79 MEN1 (0.53) CYP3A4ALDH1A1TSHRTAAR1LMNA
SCHEMBL10953000 0.79 HPGD (0.46) TSHRTAAR1ADRA2AADRA2BADRA2C
SCHEMBL3385419 0.79 MEN1 (0.54) CYP3A4ALDH1A1TAAR1LMNAPTGS1
SCHEMBL11660485 0.79 TAAR1 (0.42) TSHRTAAR1CYP17A1CYP11B1CYP11B2
SCHEMBL20738474 0.79 MEN1 (0.61) ALDH1A1TDP1TAAR1GFERADRA1D
SCHEMBL3236567 0.79 HPGD (0.53) TAAR1LMNAPTGS1PTGS2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024020164-A2 GLUCOCORTICOID RECEPTOR AGONISTS AND CONJUGATES THEREOF FIREFLY BIO, INC. (US) 2024-01-25 WO disclosed
EP-0353032-B1 1,5-BENZOTHIAZEPINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CARDIOVASCULAR DISORDERS Sankyo Company Limited (JP) 1992-02-26 EP disclosed
US-5002942-A Calcium channel blockers for cardiovascular disorders SANKYO COMPANY, LIMITED (JP) 1991-03-26 US disclosed