SCHEMBL7299156

SCHEMBL7299156

CC1(C)C[C]c2c(C#N)cccc2O1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.33
TSHR P16473 1/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300717 0.81 TRPA1 (0.31) TRPA1TSHR
SCHEMBL7290538 0.77 HTR2C (0.33)
SCHEMBL7299115 0.76 PKM (0.32)
SCHEMBL7300100 0.76
SCHEMBL7298705 0.76 HTR2C (0.32)
SCHEMBL7292477 0.75 TSHR (0.32) TRPA1TSHRKDM4EALDH1A1
SCHEMBL7298538 0.73 KDM4E (0.33) KDM4EALDH1A1
SCHEMBL7298521 0.72 KMT2A (0.32)
SCHEMBL7299153 0.70 TSHR (0.32) TRPA1TSHR
SCHEMBL7300190 0.69 TRPA1 (0.36) TRPA1TSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260444-A Cardiovascular, hypotensive WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
US-5208245-A Hypotensive agents WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-05-04 US disclosed
EP-0460418-A2 Novel Dihydropyridine derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-12-11 EP disclosed