SCHEMBL7299772

SCHEMBL7299772

CN(C)CCCCCNC(=O)CC(C=O)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.49
HDAC1 Q13547 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
KMT2A Q03164 1/20 0.48
HTT P42858 2/20 0.43
TRPV1 Q8NER1 1/20 0.42
CASP1 P29466 1/20 0.42
PKM P14618 1/20 0.42
APP P05067 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294460 0.95 ALOX15 (0.54) ALOX15HDAC1HDAC2HDAC8HDAC6
SCHEMBL7299907 0.77 ALOX15 (0.46) ALOX15HTTCASP1
SCHEMBL7319434 0.72 NPC1 (0.49) KMT2A
SCHEMBL10587659 0.72 HTR2A (0.47) ALDH1A1KMT2ASIGMAR1
SCHEMBL13196414 0.71 SIGMAR1 (0.59) HDAC1HDAC2HDAC8HDAC6ALDH1A1
SCHEMBL1915970 0.70 CPA3 (0.56) PKM
SCHEMBL8895410 0.69 LAP3 (0.50) PKM
SCHEMBL902140 0.69 ABCB1 (0.47) ALDH1A1KMT2A
SCHEMBL7293697 0.69 LMNA (0.55) KMT2A
SCHEMBL22170874 0.68 ALDH1A1 (0.44) HDAC1HDAC2HDAC8HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5401722-A Peptide analogues MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-03-28 US disclosed
EP-0501280-A2 Renin-inhibiting peptide analogues MERCK PATENT GmbH (DE) 1992-09-02 EP disclosed
EP-0446485-A2 Peptide analogues with renininhibiting activity MERCK PATENT GmbH (DE) 1991-09-18 EP disclosed
EP-0339483-A2 Renin inhbiting amino-acid derivatives MERCK PATENT GmbH (DE) 1989-11-02 EP disclosed