SCHEMBL7301518

SCHEMBL7301518

COc1ccc(C[C@H](NC(=O)N(C)CCc2ccccc2)C(=O)O)cc1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.65
FPR2 P25090 1/20 0.59
LPAR1 Q92633 1/20 0.53
NPY5R Q15761 1/20 0.52
ALDH1A1 P00352 2/20 0.51
ALOX15 P16050 1/20 0.51
MMP3 P08254 1/20 0.51
ALOX5 P09917 2/20 0.50
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
OPRK1 P41145 1/20 0.49
CA2 P00918 1/20 0.48
PPARG P37231 1/20 0.48
PPARA Q07869 1/20 0.48
LDHA P00338 1/20 0.48
ITGA4 P13612 1/20 0.48
ITGB7 P26010 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7292751 0.92 KMT2A (0.55) KMT2AFPR2NPY5RALDH1A1MMP3
SCHEMBL10534728 0.87 FPR2 (0.53) KMT2AFPR2ALDH1A1ALOX15CA2
SCHEMBL7305859 0.86 KMT2A (0.52) KMT2AFPR2ALDH1A1OPRD1PPARG
SCHEMBL6897944 0.85 KMT2A (0.61) KMT2AFPR2LPAR1ALDH1A1ALOX15
SCHEMBL9834187 0.82 FPR2 (0.59) KMT2AFPR2ALDH1A1ALOX15CA2
SCHEMBL7412226 0.82 KMT2A (0.46) KMT2AFPR2LPAR1NPY5RALDH1A1
SCHEMBL7301298 0.82 KMT2A (0.48) KMT2AFPR2ALDH1A1ALOX15CA2
SCHEMBL6895655 0.80 ITGA4 (0.54) ITGA4ITGB7
SCHEMBL7431334 0.79 KMT2A (0.50) KMT2AFPR2ALDH1A1ALOX15CA2
SCHEMBL5189503 0.79 FPR2 (0.68) KMT2AFPR2ALDH1A1ALOX15LDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258362-A Enzyme inhibitors, amides with oxetane ring ABBOTT LABORATORIES (US) 1993-11-02 US disclosed
WO-1992022313-A1 RENIN INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-12-23 WO disclosed
WO-1989010751-A1 FUNCTIONALIZED PEPTIDYL AMINODIOLS AND -TRIOLS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed
EP-0341602-A2 Renin-inhibiting functionalized peptidyl aminodiols and - triols ABBOTT LABORATORIES (US) 1989-11-15 EP disclosed