SCHEMBL7301718

SCHEMBL7301718

CS(=O)(=O)NCCN1CCC(Cn2cc(C(=O)O)c3ccccc32)CC1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 4/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2C9 P11712 1/20 0.62
ALOX15 P16050 1/20 0.62
NFKB1 P19838 1/20 0.62
PMP22 Q01453 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
KCNH2 Q12809 2/20 0.51
CNR1 P21554 5/20 0.49
PLK1 P53350 3/20 0.46
CNR2 P34972 2/20 0.45
KDM1A O60341 1/20 0.45
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4294889 0.91 HTR4 (0.61) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7305753 0.87 CNR1 (0.52) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7305923 0.87 CNR1 (0.50) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7331887 0.82 HRH2 (0.54) CNR1PLK1CNR2
SCHEMBL9344560 0.82 CNR1 (0.62) CNR1PLK1CNR2
SCHEMBL7308948 0.80 HTR4 (0.49) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL9704182 0.79 HTR4 (0.63) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7291968 0.79 CNR1 (0.62) NPSR1CNR1PLK1CNR2
SCHEMBL7300816 0.77 HTR4 (0.54) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL24437217 0.77 CNR1 (0.66) NPSR1CNR1PLK1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP claimed