SCHEMBL7308948

SCHEMBL7308948

O=C(O)c1cn(CCC2CCN(CCNS(=O)(=O)c3ccccc3)CC2)c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX15 P16050 1/20 0.49
NFKB1 P19838 1/20 0.49
PMP22 Q01453 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
KDM1A O60341 1/20 0.46
CNR2 P34972 5/20 0.45
CNR1 P21554 3/20 0.45
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
PLK1 P53350 3/20 0.42
ALDH1A1 P00352 1/20 0.42
HRH2 P25021 1/20 0.42
HTR7 P34969 1/20 0.42
P2RX7 Q99572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4294889 0.89 HTR4 (0.61) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7301718 0.80 HTR4 (0.62) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7310095 0.79 CNR2 (0.47) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7300971 0.77 HTR4 (0.81) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7308950 0.75 KDM1A (0.46) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL9543051 0.73 CNR2 (0.52) CNR2CNR1HRH2
SCHEMBL3886047 0.73 KDM1A (0.61) KDM1AALDH1A1HTR7
SCHEMBL12643110 0.70 CNR2 (0.69) CNR2CNR1PLK1ALDH1A1
SCHEMBL19048139 0.70 KDM1A (0.61) KDM1AALDH1A1HTR7
SCHEMBL7331887 0.70 HRH2 (0.54) CNR2CNR1PLK1HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP claimed