SCHEMBL7305753

SCHEMBL7305753

Cc1ccc2c(c1)c(C(=O)O)cn2CC1CCN(CCNS(C)(=O)=O)CC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.52
HTR4 Q13639 5/20 0.50
CYP2C9 P11712 2/20 0.50
CYP1A2 P05177 1/20 0.50
ALOX15 P16050 1/20 0.50
NFKB1 P19838 1/20 0.50
PMP22 Q01453 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
KCNH2 Q12809 2/20 0.42
ICMT O60725 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
GSK3B P49841 1/20 0.40
CNR2 P34972 3/20 0.39
KDM1A O60341 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7305923 0.90 CNR1 (0.50) CNR1HTR4CYP2C9CYP1A2ALOX15
SCHEMBL7301718 0.87 HTR4 (0.62) CNR1HTR4CYP2C9CYP1A2ALOX15
SCHEMBL4294889 0.79 HTR4 (0.61) CNR1HTR4CYP2C9CYP1A2ALOX15
SCHEMBL7302781 0.78 HTR4 (0.45) HTR4CYP2C9CYP1A2ALOX15NFKB1
SCHEMBL9703208 0.77 HTR4 (0.61) HTR4CYP2C9CYP1A2ALOX15NFKB1
SCHEMBL9703205 0.76 HTR4 (0.52) HTR4CYP2C9CYP1A2ALOX15NFKB1
SCHEMBL7359270 0.71 CNR1 (0.43) CNR1ICMTCNR2
SCHEMBL7313709 0.70 CYP2C9 (0.53) HTR4CYP2C9CYP1A2ALOX15NFKB1
SCHEMBL7300888 0.70 HTR4 (0.77) HTR4CYP2C9CYP1A2ALOX15NFKB1
SCHEMBL7291933 0.70 HTR4 (0.61) HTR4CYP2C9CYP1A2ALOX15NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP claimed