SCHEMBL7302420

SCHEMBL7302420

COCCn1nc(-c2ccc(O)cc2)oc1=O

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
MAOB P27338 2/20 0.45
NOTUM Q6P988 1/20 0.42
MTOR P42345 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9424210 0.79 MAOB (0.57) MAOBNOTUM
SCHEMBL12377828 0.77 GRIN1 (0.46) GAANOTUMGRIN1GRIN2B
SCHEMBL7298728 0.76 MAOB (0.42) GAAMAOB
SCHEMBL7300033 0.75 MAOB (0.43) GAAMAOBGRIN1GRIN2B
SCHEMBL13863022 0.71 ALDH1A1 (0.35)
SCHEMBL7302416 0.70 NOTUM (0.40) GAANOTUM
SCHEMBL11857867 0.68 FAAH (0.46)
SCHEMBL10703697 0.65 KDM4E (0.51) GAAMAOBGRIN1GRIN2B
SCHEMBL11869259 0.64 TDP1 (0.44) GAA
SCHEMBL10437798 0.64 MAOB (0.46) GAAMAOBNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655445-B1 1,3,4-oxadiazol-2(3H)-one Derivates, their preparation and their use as monoamine oxidase inhibitors SYNTHELABO (FR) 1997-08-27 EP disclosed
US-5525619-A INHIBITORS OF MONOAMINE OXIDASE B SYNTHELABO (FR) 1996-06-11 US disclosed
EP-0655445-A1 1,3,4-oxadiazol-2(3H)-one Derivates, their preparation and their use as monoamine oxidase inhibitors SYNTHELABO (FR) 1995-05-31 EP disclosed