SCHEMBL7302447

SCHEMBL7302447

CCOC(=O)N(CCCCN1CC=C(c2ccccc2)CC1)c1cccc(F)c1C(=O)OC

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
DRD3 P35462 1/20 0.40
SIGMAR1 Q99720 4/20 0.39
KDM4E B2RXH2 3/20 0.39
HTR7 P34969 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
HTR1A P08908 2/20 0.38
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297468 0.92 DRD3 (0.41) PARP1DRD3SIGMAR1KDM4EHTR7
SCHEMBL7301503 0.90 HTR7 (0.43) PARP1DRD3SIGMAR1KDM4EHTR7
SCHEMBL7359856 0.90 KDM4E (0.44) PARP1DRD3SIGMAR1KDM4EHTR7
SCHEMBL7310797 0.87 DRD3 (0.38) DRD3SIGMAR1KDM4EHTR7ALDH1A1
SCHEMBL7308008 0.85 SIGMAR1 (0.42) PARP1DRD3SIGMAR1KDM4EHTR7
SCHEMBL7307713 0.85 HTR7 (0.44) PARP1DRD3SIGMAR1KDM4EHTR7
SCHEMBL7310638 0.84 KDM4E (0.43) PARP1SIGMAR1KDM4EHTR7ALDH1A1
SCHEMBL7307166 0.83 KDM4E (0.43) PARP1SIGMAR1KDM4EHTR7ALDH1A1
SCHEMBL7360979 0.82 DRD3 (0.44) PARP1DRD3SIGMAR1KDM4EHTR7
SCHEMBL7300303 0.81 HTR1A (0.46) PARP1DRD3SIGMAR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304560-A Treating CNS disorders; dopamine receptor antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-19 US disclosed
EP-0481342-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed