SCHEMBL7307896

SCHEMBL7307896

COC(=O)CN1CCN(CC2CN(C3CCN(C)CC3)C(=O)O2)CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 5/20 0.46
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
SIGMAR1 Q99720 8/20 0.34
HSD17B10 Q99714 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32
CCR8 P51685 1/20 0.32
OPRL1 P41146 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311678 0.90 HTR2B (0.45) HTR2BITGB3ITGA2BSIGMAR1HSD17B10
SCHEMBL7311014 0.88 HTR2B (0.43) HTR2BITGB3ITGA2BSIGMAR1HSD17B10
SCHEMBL7302525 0.88 HTR2B (0.48) HTR2BITGB3ITGA2BSIGMAR1HRH3
SCHEMBL7313313 0.88 HTR2B (0.45) HTR2BITGB3ITGA2BSIGMAR1OPRL1
SCHEMBL7310299 0.87 HTR2B (0.51) HTR2BITGB3ITGA2BSIGMAR1HSD17B10
SCHEMBL7318339 0.86 ITGB3 (0.45) HTR2BITGB3ITGA2BSIGMAR1OPRL1
SCHEMBL7309068 0.84 HTR2B (0.41) HTR2BITGB3ITGA2B
SCHEMBL7303558 0.84 HTR2B (0.52) HTR2BITGB3ITGA2BSIGMAR1CCR8
SCHEMBL7305444 0.81 HTR2B (0.50) HTR2BSIGMAR1HSD17B10
SCHEMBL7313685 0.81 ITGB3 (0.42) HTR2BITGB3ITGA2BSIGMAR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed