SCHEMBL7302709

SCHEMBL7302709

N=C(N)c1ccc(S(=O)(=O)NCC(O)c2ccc(OCC(=O)O)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.49
ITGA2B P08514 3/20 0.49
TBXA2R P21731 1/20 0.46
TBXAS1 P24557 1/20 0.46
ALDH1A1 P00352 2/20 0.45
TMPRSS6 Q8IU80 4/20 0.43
POLB P06746 1/20 0.43
PLAU P00749 1/20 0.43
HPN P05981 1/20 0.43
IDO1 P14902 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PDK1 Q15118 1/20 0.42
PDK2 Q15119 1/20 0.42
PDK3 Q15120 1/20 0.42
PDK4 Q16654 1/20 0.42
F2 P00734 2/20 0.42
TSHR P16473 1/20 0.41
F10 P00742 1/20 0.41
PRSS1 P07477 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301011 0.89 POLB (0.57) ALDH1A1POLBPLAUHPNHSP90AA1
Hydrochloric Acid SCHEMBL9265744 0.89 POLB (0.56) ALDH1A1TMPRSS6POLBPLAUHPN
SCHEMBL9778021 0.85 TBXA2R (0.62) TBXA2RTBXAS1ALDH1A1HSP90AA1HSP90AB1
SCHEMBL9777989 0.84 TBXA2R (0.49) TBXA2RTBXAS1ALDH1A1IDO1HSP90AA1
SCHEMBL9778015 0.84 MMP2 (0.49) TBXA2RTBXAS1ALDH1A1IDO1HSP90AA1
SCHEMBL7302514 0.83 ITGB3 (0.54) ITGB3ITGA2BTBXA2RTBXAS1ALDH1A1
SCHEMBL7298011 0.82 ITGB3 (0.57) ITGB3ITGA2BALDH1A1TSHRF10
SCHEMBL7566223 0.81 TMPRSS6 (0.48) ALDH1A1TMPRSS6PLAUHPNF2
SCHEMBL7566215 0.81 TMPRSS6 (0.48) TMPRSS6PLAUHPNF2F10
SCHEMBL7292860 0.80 TBXA2R (0.72) ITGB3ITGA2BTBXA2RTBXAS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP claimed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US claimed
US-5399585-A Anitcoagulants, antiinflammatory, antitumor HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP disclosed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US disclosed
US-5084466-A Anticoagulants, antiinflammatory agents, atheriosclerosis and antitumor agents HOFFMANN-LA ROCHE INC. (US) 1992-01-28 US disclosed