SCHEMBL7303110

SCHEMBL7303110

Cc1ccc(-c2ccccc2C(=O)NC(C)(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
ALOX5AP P20292 2/20 0.51
FEN1 P39748 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.48
ALDH1A1 P00352 4/20 0.47
TSHR P16473 1/20 0.47
CHRNB2 P17787 2/20 0.46
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
CHRNA4 P43681 2/20 0.46
HDAC7 Q8WUI4 1/20 0.45
LMNA P02545 2/20 0.43
SLC6A3 Q01959 3/20 0.43
SLC6A4 P31645 2/20 0.43
ABCB1 P08183 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13701698 0.88 CHRNB2 (0.59) MAPTMEN1KMT2AALOX5APFEN1
SCHEMBL9383059 0.82 ALOX5AP (0.56) MAPTMEN1KMT2AALOX5APFEN1
SCHEMBL7305639 0.82 MAPT (0.49) MAPTMEN1KMT2AALOX5APFEN1
SCHEMBL13845096 0.81 HDAC7 (0.66) L3MBTL1ALDH1A1CHRNB2CHRNB4CHRNA3
SCHEMBL9378163 0.81 ALOX5AP (0.52) MAPTMEN1KMT2AALOX5APFEN1
SCHEMBL3491462 0.80 CTSD (0.53) MAPTL3MBTL1ALDH1A1CHRNB2CHRNB4
SCHEMBL7016057 0.80 L3MBTL1 (0.50) MEN1KMT2AL3MBTL1ALDH1A1CHRNB2
SCHEMBL6748722 0.78 MAPT (0.61) MAPTMEN1KMT2AL3MBTL1ALDH1A1
SCHEMBL13475431 0.77 RAB9A (0.64) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL7007988 0.77 L3MBTL1 (0.48) MEN1KMT2AL3MBTL1ALDH1A1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0503785-B1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP disclosed
EP-0545912-B1 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
EP-0545912-A2 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1993-06-09 EP disclosed
EP-0503785-A1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1992-09-16 EP disclosed