SCHEMBL7303201

SCHEMBL7303201

CN1C2CCCC1CC(NC(=O)Cc1cc3ccccc3[nH]1)C2

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR6 O00574 1/20 0.55
VCP P55072 1/20 0.47
NLRP3 Q96P20 1/20 0.46
GID4 Q8IVV7 1/20 0.46
HTR3E A5X5Y0 2/20 0.45
HTR3B O95264 2/20 0.45
HTR3A P46098 2/20 0.45
HTR3D Q70Z44 2/20 0.45
HTR3C Q8WXA8 2/20 0.45
GSK3B P49841 1/20 0.44
SLC22A2 O15244 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA4 P43681 1/20 0.44
KCNH2 Q12809 1/20 0.44
SLC47A1 Q96FL8 1/20 0.44
AVPR1A P37288 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23251146 0.82 HTR3A (0.52) CXCR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL8102814 0.81 VCP (0.50) CXCR6VCPHTR3EHTR3BHTR3A
SCHEMBL9876385 0.76 HTR3A (0.50) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7448002 0.76 HRH3 (0.48) VCP
SCHEMBL34468335 0.75 KDR (0.52) NLRP3GID4GSK3B
SCHEMBL7296680 0.74 HRH3 (0.52) CXCR6VCPHTR3EHTR3BHTR3A
SCHEMBL18876541 0.74 NLRP3 (0.56) NLRP3GSK3B
SCHEMBL17327742 0.72 NLRP3 (0.60) NLRP3GSK3B
Maleic Acid SCHEMBL7333919 0.72 KDM4E (0.49) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8947376 0.70 HTR3A (0.64) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0385722-B1 Tricyclic lactam derivatives and pharmaceutical compositions containing them GLAXO GROUP LTD (GB) 1995-04-19 EP disclosed