SCHEMBL7305151

SCHEMBL7305151

CN1CCN(CCN2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAOA P21397 1/20 0.32
HRH3 Q9Y5N1 1/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314320 0.88 MAPK1 (0.37) MAPK1L3MBTL1
SCHEMBL7305380 0.84 MAPK1 (0.46) MAPK1L3MBTL1
SCHEMBL7306386 0.84 MAPK1 (0.47) MAPK1L3MBTL1DRD2DRD3
SCHEMBL7316915 0.84 MAPK1 (0.45) MAPK1L3MBTL1
SCHEMBL9230345 0.82 MAPK1 (0.49) MAPK1L3MBTL1MAOADRD2DRD3
SCHEMBL7236582 0.82 CHRM2 (0.38)
SCHEMBL7310863 0.81 MAPK1 (0.40) MAPK1L3MBTL1MAOAHRH3DRD2
SCHEMBL7229039 0.81 MAPK1 (0.36) MAPK1L3MBTL1MAOA
SCHEMBL7313654 0.81 MAPK1 (0.41) MAPK1L3MBTL1MAOA
SCHEMBL8858148 0.80 ITGB3 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed