SCHEMBL7306128

SCHEMBL7306128

[O]c1c(C(Cl)Cl)cccc1C(Cl)Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
PGK1 P00558 2/20 0.34
PGK2 P07205 2/20 0.34
CYP1A2 P05177 3/20 0.32
CYP3A4 P08684 2/20 0.32
LMNA P02545 2/20 0.32
FAAH O00519 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
GABRA1 P14867 1/20 0.32
HPGD P15428 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR2C P28335 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3785333 0.76 TSHR (0.50) TSHRCYP1A2CYP3A4LMNAFAAH
SCHEMBL6820234 0.75 CYP1A2 (0.45) TSHRPGK1PGK2CYP1A2CYP3A4
SCHEMBL7306133 0.73 GABRA1 (0.55) TSHRPGK1PGK2CYP1A2CYP3A4
SCHEMBL8728826 0.73 TSHR (0.35) TSHRCYP1A2CYP3A4LMNAFAAH
SCHEMBL7305908 0.71 ALDH1A1 (0.44) TSHRCYP1A2CYP3A4HPGDHIF1A
SCHEMBL3911665 0.69 TSHR (0.38) TSHR
SCHEMBL1872442 0.69 CYP1A2 (0.58) TSHRCYP1A2CYP3A4LMNASLC6A2
SCHEMBL199413 0.69 GABRA1 (0.57) TSHRCYP1A2CYP3A4LMNAFAAH
SCHEMBL5850205 0.67 GABRA1 (0.33) TSHRGABRA1GABRG2GABRB3
SCHEMBL5589720 0.67 ALDH1A1 (0.52) TSHRCYP1A2CYP3A4LMNAFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed