SCHEMBL8728826

SCHEMBL8728826

[CH]c1c(C(Cl)Cl)cccc1C(Cl)Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
CYP1A2 P05177 3/20 0.31
CYP3A4 P08684 2/20 0.31
FAAH O00519 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
LMNA P02545 1/20 0.31
GABRA1 P14867 1/20 0.31
HPGD P15428 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRG2 P18507 1/20 0.31
PTGS1 P23219 1/20 0.31
SLC6A2 P23975 1/20 0.31
HTR2C P28335 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
HTR2B P41595 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3785333 0.74 TSHR (0.50) TSHRCYP1A2CYP3A4FAAHCA1
SCHEMBL6820234 0.73 CYP1A2 (0.45) TSHRCYP1A2CYP3A4FAAHCA1
SCHEMBL7306128 0.73 TSHR (0.36) TSHRCYP1A2CYP3A4FAAHCA1
SCHEMBL7306133 0.71 GABRA1 (0.55) TSHRCYP1A2CYP3A4FAAHCA1
SCHEMBL8724963 0.69 TSHR (0.33) TSHR
SCHEMBL1872442 0.67 CYP1A2 (0.58) TSHRCYP1A2CYP3A4LMNASLC6A2
SCHEMBL2418565 0.66 P2RX7 (0.43) TSHRCYP1A2CYP3A4LMNACYP2A6
SCHEMBL10493638 0.65 TSHR (0.36) TSHR
SCHEMBL5850205 0.65 GABRA1 (0.33) TSHRGABRA1GABRG2GABRB3
SCHEMBL1845725 0.65 TSHR (0.36) TSHRCYP3A4LMNASLC6A2HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609058-B1 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO CO (JP) 1998-12-09 EP disclosed
US-5491167-A INHIBITORS OF CHOLESTEROL BIOSYNTHESIS SANKYO COMPANY, LIMITED (JP) 1996-02-13 US disclosed
EP-0609058-A2 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO COMPANY LIMITED (JP) 1994-08-03 EP disclosed