SCHEMBL7308175

SCHEMBL7308175

NC(=S)Oc1ccc(Cl)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.46
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
IDO1 P14902 2/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CHRNA3 P32297 1/20 0.39
KMO O15229 1/20 0.39
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP3A5 P20815 1/20 0.38
CYP2C19 P33261 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7165371 0.81 HSP90AA1 (0.47) HSP90AA1GLAGAAMAPTIDO1
SCHEMBL11627822 0.79 HSP90AA1 (0.46) HSP90AA1HTR3EHTR3BHTR3AHTR3D
SCHEMBL23753577 0.79 MEN1 (0.57) HSP90AA1HTR3EHTR3BHTR3AHTR3D
SCHEMBL27617217 0.76 MAOA (0.43) MAPTHTR3EHTR3BHTR3AHTR3D
SCHEMBL9255310 0.74 HSP90AA1 (0.48) HSP90AA1SLC6A2SLC6A4SLC6A3CHRNA3
Fluoride SCHEMBL28396424 0.74 MAOA (0.41) MAPTHTR3EHTR3BHTR3AHTR3D
SCHEMBL7659746 0.73 WDR5 (0.51) GAAMAPTHTR3EHTR3BHTR3A
SCHEMBL1587868 0.72 KDM4E (0.47) HSP90AA1SLC6A2SLC6A4SLC6A3CHRNA3
SCHEMBL9666256 0.71 TDP1 (0.52) GAAMAPTHTR3EHTR3BHTR3A
SCHEMBL9485744 0.71 KMO (0.46) HSP90AA1MAPTSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5674864-A ANALGESICS; ENDOPEPTIDASE AND ENKEPHALINASE INHIBITORS; CARDIOTONIC, PSYCHOTROPIC AND HYPERTENSIVE AGENTS ROUSSEL UCLAF (FR) 1997-10-07 US disclosed
EP-0465369-B1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1994-04-13 EP disclosed
US-5190974-A Analgesics ROUSSEL UCLAF (FR) 1993-03-02 US disclosed