SCHEMBL7308323

SCHEMBL7308323

CNc1ccc(C2=NOC(c3ccccc3)N2)cc1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
P2RX7 Q99572 2/20 0.33
APP P05067 2/20 0.33
MEN1 O00255 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM1A O60341 1/20 0.33
NISCH Q9Y2I1 1/20 0.31
KIF11 P52732 1/20 0.30
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313645 0.80 HSD17B10 (0.39) TSHRP2RX7MEN1GLAKMT2A
SCHEMBL7638239 0.79 MEN1 (0.43) P2RX7MEN1KMT2A
SCHEMBL7304049 0.76 BCHE (0.40)
SCHEMBL24181414 0.72 GPR88 (0.31)
SCHEMBL15952330 0.72 CYP2A6 (0.42) P2RX7
SCHEMBL23019900 0.68 ALDH1A1 (0.47) MEN1GAAKMT2A
SCHEMBL18507295 0.68 KMO (0.47) GAA
SCHEMBL15951872 0.65 KMT2A (0.38) TSHRMEN1GAAKMT2ANISCH
SCHEMBL223709 0.65 TSHR (0.68) TSHRAPPMEN1GLAGAA
SCHEMBL17283460 0.65 TSHR (0.68) TSHRAPPMEN1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed