SCHEMBL7308356

SCHEMBL7308356

CCCCc1nc(C(C)(C)O)c(C(=O)OC)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.36
TLR7 Q9NYK1 2/20 0.36
GPR84 Q9NQS5 5/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
PARP1 P09874 1/20 0.33
LMNA P02545 1/20 0.33
TUBB4A P04350 1/20 0.33
CYP1A2 P05177 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2121837 0.92 HCRTR1 (0.35) TLR7HCRTR1HCRTR2ALDH1A1MAPK1
SCHEMBL7298547 0.88 ALDH1A1 (0.40) ALDH1A1MAPK1LMNACYP1A2CYP2D6
SCHEMBL833 0.81 GPR84 (0.37) GPR84NPC1RAB9AALDH1A1MAPK1
SCHEMBL7883601 0.81 PDE2A (0.33) NPC1RAB9AMAPK1MAPT
SCHEMBL27334926 0.80 GPR84 (0.41) GPR84NPC1RAB9AALDH1A1MAPK1
SCHEMBL7303318 0.80 NPSR1 (0.41) GPR84NPC1RAB9AALDH1A1MAPK1
SCHEMBL2123507 0.79 LMNA (0.41) GPR84NPC1RAB9AALDH1A1MAPK1
SCHEMBL27446651 0.79 ALDH1A1 (0.33) ALDH1A1
SCHEMBL987234 0.79 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL9873189 0.78 GPR84 (0.37) TLR8TLR7GPR84NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1101384-C Process for preparing 1-biphenylmethylimidazole derivatives SANKYO CO (JP) 2003-02-12 CN disclosed
EP-0503785-B1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP disclosed
CN-1045770-C Process for preparing 1-biphenylmethylimidazole derivatives SANKYO CO (JP) 1999-10-20 CN disclosed
CN-1189490-A Process for preparing 1-biphenylmethylimidazole derivatives SANKYO CO (JP) 1998-08-05 CN disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
CN-1065063-A 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1992-10-07 CN disclosed
EP-0503785-A1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1992-09-16 EP disclosed