SCHEMBL7310501

SCHEMBL7310501

FC(F)(F)C1Cc2ccccc2C=N1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.37
TRPA1 O75762 1/20 0.35
IDO1 P14902 2/20 0.31
CYP19A1 P11511 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11781894 0.98 PNMT (0.36) PNMTTRPA1IDO1
SCHEMBL22244282 0.81 TRPA1 (0.35) TRPA1IDO1CYP19A1CYP11B1CYP11B2
SCHEMBL18464841 0.75 TRPA1 (0.38) TRPA1IDO1CYP19A1CYP11B1CYP11B2
SCHEMBL31303677 0.71 NOS3 (0.43) TRPA1IDO1CYP19A1CYP11B1CYP11B2
SCHEMBL5008439 0.71 NOS3 (0.43) TRPA1IDO1CYP19A1CYP11B1CYP11B2
SCHEMBL16930290 0.68 CYP3A4 (0.37)
SCHEMBL4130355 0.68 NOS3 (0.46) TRPA1
SCHEMBL8628901 0.67 TRPA1 (0.35) TRPA1IDO1CYP19A1CYP11B1CYP11B2
SCHEMBL3979211 0.67 TRPA1 (0.35) TRPA1IDO1CYP19A1CYP11B1CYP11B2
SCHEMBL31168159 0.67 TRPA1 (0.35) TRPA1IDO1CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617166-A Protein Kinase Inhibitor Benzolactam Compounds 大冢制药株式会社 2018-10-02 CN disclosed
US-5605926-A PROPHYLAXIS BAYER AKTIENGESELLSCHAFT (DE) 1997-02-25 US disclosed
US-5430151-A Treatment of aids, pneumonia, caprine arthritis encephalitis, leukemia and immmunodeficiency BAYER AKTIENGESELLSCHAFT (DE) 1995-07-04 US disclosed
US-5204471-A α-trifluoromethyl-substituted, saturated bicyclic amines BAYER AKTIENGESELLSCHAFT (DE) 1993-04-20 US disclosed
EP-0528242-A2 Trifluoromethyl containing pseudopeptides BAYER AG (DE) 1993-02-24 EP disclosed
EP-0527385-A1 Alpha-trifluoromethyl substituted, saturated bicyclic amines and process for their preparation BAYER AG (DE) 1993-02-17 EP disclosed
US-3956333-A BACTERICIDE STERLING DRUG INC. (US) 1976-05-11 US disclosed