SCHEMBL7311963

SCHEMBL7311963

CC(COc1ccc2c(c1)CCC(=O)N2)Cc1nnnn1Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 12/20 0.53
MAOB P27338 12/20 0.53
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46
MEN1 O00255 1/20 0.46
ABCC4 O15439 1/20 0.46
CACNA1F O60840 1/20 0.46
ABCB11 O95342 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
THPO P40225 1/20 0.46
OPRK1 P41145 1/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309846 0.84 MAOA (0.69) MAOAMAOBPDE3BPDE3AMEN1
SCHEMBL7306908 0.79 PDE3B (0.71) MAOAMAOBPDE3BPDE3AMEN1
SCHEMBL7313754 0.79 MAOB (0.65) MAOAMAOBDRD2
SCHEMBL7310807 0.77 MAOB (0.69) MAOAMAOBPDE3BPDE3AMEN1
SCHEMBL7316158 0.77 ALDH1A1 (0.47) MAOBPDE3BPDE3AMEN1ALDH1A1
SCHEMBL7306011 0.73 PDE3B (0.65) MAOAMAOBPDE3BPDE3AMEN1
SCHEMBL10572504 0.71 KCNH2 (0.70) MAOAMAOBALDH1A1LMNACYP2C9
SCHEMBL2236580 0.71 MAOB (1.00) MAOAMAOB
SCHEMBL7309989 0.70 MAOA (0.64) MAOAMAOBPDE3BPDE3AMEN1
SCHEMBL7317621 0.69 ALDH1A1 (0.38) PDE3BPDE3AMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4277479-A ANTI-ASTHMATIC, HYPOTENSIVE, ANTI-ULCER, ANTIINFLAMMATORY, VASODILATION, ENZYME INHIBITORS, ANTICOAGULANTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1981-07-07 US disclosed