SCHEMBL7316540

SCHEMBL7316540

COC(=O)c1cccc(C=O)c1NS(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.62
TCF4 P15884 1/20 0.54
CTNNB1 P35222 1/20 0.54
FFAR4 Q5NUL3 3/20 0.53
HPGD P15428 3/20 0.51
ALDH1A1 P00352 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
HTT P42858 2/20 0.51
TP53 P04637 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CYP19A1 P11511 1/20 0.50
TSHR P16473 3/20 0.49
KDM4E B2RXH2 1/20 0.48
USP2 O75604 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ELANE P08246 1/20 0.47
PRTN3 P24158 1/20 0.47
CYP2C9 P11712 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CYTH2 Q99418 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324918 0.90 LMNA (0.51) LMNATCF4CTNNB1FFAR4HPGD
SCHEMBL7324979 0.83 LMNA (0.67) LMNATCF4CTNNB1FFAR4HPGD
SCHEMBL5159892 0.83 FFAR4 (0.74) LMNATCF4CTNNB1FFAR4HPGD
SCHEMBL7312055 0.82 LMNA (0.65) LMNATCF4CTNNB1FFAR4HPGD
SCHEMBL7322570 0.82 LMNA (0.65) LMNATCF4CTNNB1FFAR4HPGD
SCHEMBL5158052 0.78 LMNA (0.79) LMNAFFAR4HPGDALDH1A1L3MBTL1
SCHEMBL7322457 0.76 MMP2 (0.40) LMNATCF4CTNNB1HPGDALDH1A1
SCHEMBL7325109 0.75 MMP1 (0.49) LMNAHPGDALDH1A1L3MBTL1HTT
SCHEMBL7316215 0.75 MMP13 (0.41) LMNAHPGDALDH1A1SMN1; SMN2KDM4E
SCHEMBL7506222 0.75 LMNA (0.39) LMNATCF4CTNNB1HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0938471-B1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID CO (US) 2001-12-12 EP disclosed
EP-0938471-A1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS American Cyanamid Company (US) 1999-09-01 EP disclosed
US-5929097-A INHIBIT TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME AMERICAN CYANAMID COMPANY (US) 1999-07-27 US disclosed
WO-1998016503-A2 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1998-04-23 WO disclosed