SCHEMBL7316693

SCHEMBL7316693

O=C(O)N[C@@H](CC1CCCCC1)[C@@H](O)c1nccs1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.43
EPHX2 P34913 1/20 0.42
CNR2 P34972 4/20 0.41
CTSK P43235 1/20 0.41
GCK P35557 8/20 0.39
KCNH2 Q12809 1/20 0.37
MEN1 O00255 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HTT P42858 1/20 0.37
ADAM17 P78536 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7316703 1.00 POLB (0.43) POLBEPHX2CNR2CTSKGCK
SCHEMBL9705262 0.83 REN (0.46) POLBCNR2CTSKKCNH2
SCHEMBL9705257 0.83 REN (0.46) POLBCNR2CTSKKCNH2
SCHEMBL9740697 0.82 REN (0.41) CNR2CTSKGCK
SCHEMBL7424256 0.82 REN (0.41) CNR2CTSKGCK
SCHEMBL9740699 0.82 REN (0.41) CNR2CTSKGCK
SCHEMBL7269773 0.78 CTSC (0.38) POLBEPHX2CTSKGCKKCNH2
SCHEMBL7269778 0.78 CTSC (0.38) POLBEPHX2CTSKGCKKCNH2
SCHEMBL15689096 0.78 ADAM17 (0.41) TSHRADAM17
SCHEMBL7424258 0.77 CCR1 (0.40) POLBEPHX2CNR2CTSKGCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231919-B1 N-HETEROCYCLIC ALCOHOL RENIN INHIBITORS E.R. Squibb & Sons, Inc. (US) 1993-01-20 EP disclosed
US-4885292-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1989-12-05 US disclosed
EP-0231919-A2 N-Heterocyclic alcohol renin inhibitors E.R. Squibb & Sons, Inc. (US) 1987-08-12 EP disclosed