SCHEMBL7318604

SCHEMBL7318604

N=C(N)c1ccc(N2CCN(C(Oc3ccccc3)C(=O)O)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.55
ITGA2B P08514 13/20 0.55
F2 P00734 2/20 0.54
PRSS1 P07477 2/20 0.54
PRSS2 P07478 2/20 0.54
PRSS3 P35030 2/20 0.54
TMPRSS6 Q8IU80 2/20 0.54
ST14 Q9Y5Y6 2/20 0.54
GRIN2D O15399 1/20 0.50
GRIN3B O60391 1/20 0.50
GRIN1 Q05586 1/20 0.50
GRIN2A Q12879 1/20 0.50
GRIN2B Q13224 1/20 0.50
GRIN2C Q14957 1/20 0.50
GRIN3A Q8TCU5 1/20 0.50
ALOX15 P16050 2/20 0.43
PARP14 Q460N5 1/20 0.40
PARP10 Q53GL7 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696501 0.80 CYP2C9 (0.49) ITGB3ITGA2BALOX15ALDH1A1MAPT
SCHEMBL7318615 0.76 OPRD1 (0.41) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL7347645 0.73 F2 (0.58) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL2403330 0.73 F2 (1.00) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL10187743 0.73 HSD17B10 (0.49) ALOX15NPC1ALDH1A1LMNAMAPT
SCHEMBL7315288 0.71 ITGB3 (0.68) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL7782353 0.70 ITGB3 (1.00) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL6705795 0.70 LMNA (0.55) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL7317414 0.70 OPRD1 (0.47) ALDH1A1TSHRHSD17B10
SCHEMBL7439185 0.70 ITGB3 (0.52) ITGB3ITGA2BF2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843948-A Piperazinophenyl- and piperazinophenyloxycarboxylic acid derivatives, and processes and intermediates for their preparation and pharmaceutical compositions comprising them SOLVAY PHARMACEUTICALS GMBH (DE) 1998-12-01 US claimed
US-5843948-A Piperazinophenyl- and piperazinophenyloxycarboxylic acid derivatives, and processes and intermediates for their preparation and pharmaceutical compositions comprising them SOLVAY PHARMACEUTICALS GMBH (DE) 1998-12-01 US disclosed