SCHEMBL7320863

SCHEMBL7320863

Brc1cn2c(Br)cnc2c(N2CCCCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.41
TSHR P16473 4/20 0.39
SCN10A Q9Y5Y9 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 2/20 0.37
MAPT P10636 2/20 0.34
LMNA P02545 1/20 0.34
PRNP P04156 1/20 0.34
ALOX15 P16050 1/20 0.34
PPARG P37231 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NR2E3 Q9Y5X4 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
AURKA O14965 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9775094 0.86 ALDH1A1 (0.47) HTR2CTSHRALDH1A1MAPK1AURKA
SCHEMBL25598043 0.75 ADORA3 (0.50) ADORA3
SCHEMBL14536745 0.72 AURKA (0.30) AURKA
SCHEMBL10092226 0.72 ALDH1A1 (0.45) TSHRALDH1A1MAPK1AURKAKDM4E
SCHEMBL29195507 0.71 HTR2C (0.36) HTR2CSCN10A
SCHEMBL29195525 0.70 HTR2C (0.36) HTR2C
SCHEMBL2317513 0.69 CYP1A2 (0.47) TSHRALDH1A1MAPK1MAPTHSD17B10
SCHEMBL20459986 0.68 TSHR (0.42) TSHRALDH1A1MAPK1MAPTLMNA
SCHEMBL22234855 0.67 MAPT (0.49) TSHRALDH1A1MAPK1MAPTKDM4E
SCHEMBL2321134 0.67 TSHR (0.44) TSHRALDH1A1MAPK1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5028605-A Antispasmodic, bronchodilators, uterine relaxants, cardiac analeptics, neurosedatives L'UNIVERSITE DE MONTPELLIER I (FR) 1991-07-02 US disclosed
EP-0348392-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY Université Montpellier I (FR) 1990-01-03 EP disclosed
WO-1988004298-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1988-06-16 WO disclosed