SCHEMBL7325931

SCHEMBL7325931

COc1ccccc1C1(OC(C)[C@H](N)C(=O)O)c2ccccc2-c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
AKR1C3 P42330 3/20 0.39
AKR1C2 P52895 3/20 0.39
ACHE P22303 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KIF11 P52732 3/20 0.35
TACR1 P25103 1/20 0.35
PDK2 Q15119 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7325936 1.00 KMT2A (0.41) KMT2AAKR1C3AKR1C2ACHECA1
SCHEMBL7322362 0.84 ACHE (0.44) KMT2AAKR1C3AKR1C2ACHEALDH1A1
SCHEMBL7322359 0.84 ACHE (0.44) KMT2AAKR1C3AKR1C2ACHEALDH1A1
SCHEMBL7325812 0.84 KIF11 (0.38) KMT2AAKR1C3AKR1C2TDP1KIF11
SCHEMBL7325808 0.84 KIF11 (0.38) KMT2AAKR1C3AKR1C2TDP1KIF11
SCHEMBL7317362 0.84 KIF11 (0.44) KMT2AKDM4EALDH1A1HPGDTDP1
SCHEMBL7323867 0.84 KIF11 (0.44) KMT2AKDM4EALDH1A1HPGDTDP1
SCHEMBL7317367 0.84 KIF11 (0.44) KMT2AKDM4EALDH1A1HPGDTDP1
SCHEMBL7320576 0.83 KIF11 (0.38) KMT2AAKR1C3AKR1C2TSHRALDH1A1
SCHEMBL7320568 0.83 KIF11 (0.38) KMT2AAKR1C3AKR1C2TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO claimed
US-6162824-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ALLELIX NEUROSCIENCE INC. 2000-12-19 US disclosed
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO disclosed