SCHEMBL7327586

SCHEMBL7327586

O=C(O)COc1cccc(NS(=O)(=O)c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.58
ROCK2 O75116 1/20 0.56
BRAF P15056 1/20 0.56
KMT2A Q03164 3/20 0.55
FABP1 P07148 1/20 0.54
ERAP1 Q9NZ08 1/20 0.54
AR P10275 1/20 0.54
MAPT P10636 2/20 0.53
LMNA P02545 2/20 0.52
MEN1 O00255 1/20 0.52
PTPN1 P18031 2/20 0.52
IDH1 O75874 1/20 0.52
FFAR1 O14842 1/20 0.51
CDK1 P06493 1/20 0.51
CCNB1 P14635 1/20 0.51
CCNA2 P20248 1/20 0.51
CDK2 P24941 1/20 0.51
CDK7 P50613 1/20 0.51
CCNH P51946 1/20 0.51
CCNA1 P78396 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324171 0.90 NR3C1 (0.61) BRAFKMT2AARMAPTLMNA
SCHEMBL7325645 0.88 F2 (0.60) FABP1ARLMNAPTPN1FFAR1
SCHEMBL7330191 0.86 FABP1 (0.62) BRAFKMT2AFABP1ERAP1MAPT
SCHEMBL7327897 0.86 IDH1 (0.57) EPHX2ROCK2BRAFKMT2AERAP1
SCHEMBL7324870 0.84 F2 (0.59) FABP1MAPTLMNAFFAR1CDK1
SCHEMBL7335570 0.84 CYP19A1 (0.61) BRAFFABP1ARLMNAMAPK1
SCHEMBL7359983 0.84 ROCK2 (0.62) EPHX2ROCK2KMT2AMAPTLMNA
SCHEMBL9812957 0.82 CYP19A1 (0.67) KMT2AARLMNAMEN1
SCHEMBL17468424 0.82 PGR (0.65) EPHX2BRAFKMT2AERAP1AR
SCHEMBL7324125 0.81 F2 (0.60) KMT2AFABP1LMNAMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687253-B1 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1998-12-16 EP disclosed
EP-0687253-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME Roche Diagnostics GmbH (DE) 1995-12-20 EP disclosed
WO-1994020467-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1994-09-15 WO disclosed