SCHEMBL7327875

SCHEMBL7327875

CCCC(C)(Cc1c(NC(C)=O)ccc(C(=O)OC)c1O)OS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
STAT3 P40763 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
LMNA P02545 4/20 0.35
TSHR P16473 2/20 0.35
FFAR4 Q5NUL3 1/20 0.35
ESR1 P03372 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPK1 P28482 1/20 0.34
PKM P14618 2/20 0.33
CDK1 P06493 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7328711 0.91 STAT3 (0.42) KMT2ASTAT3CTDSP1SIRT5SMN1; SMN2
SCHEMBL7328403 0.79 SMN1; SMN2 (0.40) KMT2ASMN1; SMN2LMNAESR1ALDH1A1
SCHEMBL7325433 0.77 PSMD10 (0.43) KMT2ASTAT3CTDSP1SIRT5SMN1; SMN2
SCHEMBL7327836 0.74 KMT2A (0.38) KMT2ASTAT3CTDSP1SIRT5SMN1; SMN2
SCHEMBL13215874 0.68 SMN1; SMN2 (0.43) KMT2ASMN1; SMN2LMNATSHRALDH1A1
SCHEMBL6896594 0.68 ALDH1A1 (0.45) KMT2ASMN1; SMN2ALDH1A1
SCHEMBL19211610 0.67 SMN1; SMN2 (0.46) KMT2ASMN1; SMN2LMNATSHRALDH1A1
SCHEMBL7327731 0.67 CYP4A11 (0.43) KMT2ASMN1; SMN2LMNATSHRALDH1A1
SCHEMBL9868368 0.67 SMN1; SMN2 (0.43) KMT2ASMN1; SMN2LMNATSHRALDH1A1
SCHEMBL19211596 0.66 SMN1; SMN2 (0.44) KMT2ASMN1; SMN2LMNATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4924010-A GASTROINTESTINAL DISORDERS RORER PHARMACEUTICAL CORPORATION (US) 1990-05-08 US disclosed
US-4859683-A Certain benzoxepins and their pharmaceutical compositions and methods RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
US-4857517-A Quinuclidyl benzoxepins as 5-HT3 antagonists RORER PHARMACEUTICAL CORPORATION (US) 1989-08-15 US disclosed