SCHEMBL7334393

SCHEMBL7334393

CC(C)(C)C(=O)Nc1ccc(CC#N)c(OCC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP1A2 P05177 1/20 0.40
LCK P06239 1/20 0.39
CTSL P07711 1/20 0.39
PTPRC P08575 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
CTSS P25774 1/20 0.39
PTPN13 Q12923 1/20 0.39
UGCG Q16739 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339466 0.77 RXRA (0.36) CYP2C9CYP1A2UGCG
SCHEMBL7342162 0.73 MEN1 (0.39) ARL3MBTL1UGCGMAPT
SCHEMBL429691 0.72 CYP3A4 (0.49) L3MBTL1LCKCTSLPTPRCPTPN2
SCHEMBL7343829 0.70 NR1H4 (0.47) MAPT
SCHEMBL7341428 0.69 ALDH1A1 (0.41) CYP2C9CYP2C19CYP1A2MAPT
SCHEMBL1817634 0.68 CA12 (0.43) ARL3MBTL1CYP2C9CYP2C19CYP1A2
SCHEMBL7334398 0.68 L3MBTL1 (0.47) ARL3MBTL1MAPT
SCHEMBL9430893 0.67 AR (0.63) ARCYP2C19
SCHEMBL2956472 0.66 AR (0.44) ARL3MBTL1
SCHEMBL5404961 0.65 CYP2C9 (0.60) ARL3MBTL1CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
US-5968938-A Piperazine oxytocin receptor antagonists MERCK & CO., INC. (US) 1999-10-19 US disclosed