SCHEMBL7334530

SCHEMBL7334530

O=S(=O)(Cl)c1c(F)ccc(-c2c(F)cccc2F)c1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.39
PKLR P30613 1/20 0.39
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
PTGES2 Q9H7Z7 3/20 0.31
PTGS2 P35354 5/20 0.31
PTGS1 P23219 2/20 0.31
PDK2 Q15119 1/20 0.31
PDCD1LG2 Q9BQ51 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
TTR P02766 1/20 0.31
CES2 O00748 1/20 0.31
BCHE P06276 1/20 0.31
CES1 P23141 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
HTR5A P47898 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2238428 0.80 ACLY (0.38) PTGS2PTGS1ALDH1A1HSD17B10TDP1
SCHEMBL532887 0.80 PKM (0.50) PKMPKLRPTGES2CES2BCHE
SCHEMBL30986771 0.78 CA1 (0.39) PKMPKLRCA1CA2CA7
SCHEMBL3523738 0.78 CA1 (0.39) PKMPKLRCA1CA2CA7
SCHEMBL31454807 0.72 PKM (0.35) PKMPKLRCA1CA2CA7
SCHEMBL4537200 0.72 PKM (0.48) PKMPKLRALDH1A1TDP1
SCHEMBL19858507 0.71 PKM (0.42) PKMPKLRCA1CA2CA9
SCHEMBL22146034 0.71 PTGS2 (0.34) PKMPKLRCA1CA2CA7
SCHEMBL20560224 0.71 PKM (0.42) PKMPKLRPTGES2CES2CES1
SCHEMBL29764209 0.71 ACHE (0.44) PKMPKLRALDH1A1HSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997046207-A2 AROMATIC HETEROCYCLIC DERIVATIVES AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1997-12-11 WO disclosed
EP-0804464-A1 AROMATIC HETEROCYCLIC DERIVATIVES AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1997-11-05 EP disclosed
WO-1996018644-A1 AROMATIC HETEROCYCLIC DERIVATIVES AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1996-06-20 WO disclosed