SCHEMBL7334908

SCHEMBL7334908

Nc1cccc(NCC(=O)Nc2ccncc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.52
HDAC4 P56524 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC10 Q969S8 1/20 0.52
HDAC11 Q96DB2 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
HDAC9 Q9UKV0 1/20 0.52
HDAC5 Q9UQL6 1/20 0.52
DDX3X O00571 1/20 0.49
GRK2 P25098 9/20 0.48
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47
CDK3 Q00526 1/20 0.47
GRK3 P35626 6/20 0.47
GRK5 P34947 1/20 0.47
ALDH1A1 P00352 1/20 0.46
ROCK2 O75116 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14625936 0.82 IMPDH2 (0.55) ROCK2
SCHEMBL7334697 0.81 GRK2 (0.44) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8547667 0.79 MEN1 (0.58) HDAC1DDX3XGRK2ALDH1A1MEN1
SCHEMBL8547282 0.76 KMT2A (0.56) HDAC8HDAC6GRK2GRK3ALDH1A1
SCHEMBL3646757 0.75 ALDH1A1 (0.64) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6370197 0.75 DDX3X (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL17560624 0.75 DDX3X (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4518077 0.74 PORCN (0.64) HDAC1GRK2ALDH1A1ROCK2TAAR1
SCHEMBL10884504 0.73 DDX3X (0.55) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8549861 0.73 ALDH1A1 (0.54) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687253-B1 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1998-12-16 EP disclosed
EP-0687253-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME Roche Diagnostics GmbH (DE) 1995-12-20 EP disclosed
WO-1994020467-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1994-09-15 WO disclosed