SCHEMBL7337341

SCHEMBL7337341

CCCOc1ccc2c(c1)S(=O)(=O)N(C(C)(C)C)C2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.44
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
MAPT P10636 3/20 0.37
KMT2A Q03164 3/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 2/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PDK2 Q15119 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1369709 0.73 PTGDR2 (0.42) PTGDR2CA12CA1CA2CA7
SCHEMBL7340305 0.70 CA12 (0.50) CA12CA1CA2CA6CA5A
SCHEMBL20443155 0.68 CA2 (0.43) CA2CA9KMT2ARAB9AMEN1
SCHEMBL11579683 0.64 TOP1 (0.57) CA12CA1CA2CA6CA5A
SCHEMBL25904287 0.64 MAPK1 (0.44) CA1CA2CA7CA9CA14
SCHEMBL8545293 0.64 KMT2A (0.37) PTGDR2CA12CA1CA2CA9
SCHEMBL25920261 0.64 AOC3 (0.44) MAPTKMT2ARAB9AMEN1NPC1
SCHEMBL23051433 0.63 MAPT (0.60) MAPTKMT2ARAB9AMEN1NPC1
SCHEMBL21543709 0.63 CA12 (0.50) CA12CA1CA2CA6CA5A
SCHEMBL7284252 0.63 MAOA (0.63) CA12CA1CA2CA6CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811001-B1 BENZOTHIAZINE DIOXIDES AS ENDOTHELIN ANTAGONISTS WARNER LAMBERT CO (US) 2001-10-31 EP disclosed
WO-1996026195-A1 BENZOTHIAZINE DIOXIDES AS ENDOTHELIN ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1996-08-29 WO disclosed