SCHEMBL7337563

SCHEMBL7337563

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCC(C=O)N2CCN(C)CC2)ccc1NC(=O)c1ccccc1SCCCN

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.33
PKM P14618 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HCN1 O60741 1/20 0.32
HCN4 Q9Y3Q4 1/20 0.32
AVPR2 P30518 1/20 0.32
AVPR1A P37288 1/20 0.32
AVPR1B P47901 1/20 0.32
TP53 P04637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYP3A4 P08684 1/20 0.32
LPAR1 Q92633 1/20 0.32
ADRA1D P25100 2/20 0.32
ADRA1A P35348 2/20 0.32
ADRA1B P35368 2/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
MAP3K7 O43318 1/20 0.32
ABCB1 P08183 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7335533 0.89 ABCB1 (0.34) HCN1HCN4AVPR2AVPR1AAVPR1B
SCHEMBL7346091 0.88 HCN1 (0.35) HCN1HCN4AVPR2AVPR1AAVPR1B
SCHEMBL7342040 0.87 LMNA (0.37) MAPTALDH1A1TP53
Hydrochloric Acid SCHEMBL7778661 0.87 LMNA (0.37) MAPTALDH1A1TP53ADRA1DADRA1A
SCHEMBL7337544 0.87 AVPR2 (0.40) MAPTPKMTDP1ALDH1A1AVPR2
SCHEMBL7420333 0.87 CYP3A4 (0.34) HCN1HCN4AVPR2AVPR1AAVPR1B
SCHEMBL7337579 0.85 AVPR2 (0.34) MAPTPKMTDP1ALDH1A1AVPR2
SCHEMBL7962148 0.84 IRAK4 (0.34) HCN1HCN4AVPR2AVPR1AAVPR1B
SCHEMBL7338649 0.84 AVPR2 (0.36) MAPTAVPR2AVPR1AAVPR1BTP53
Hydrochloric Acid SCHEMBL7424661 0.84 IRAK4 (0.33) HCN1HCN4AVPR2AVPR1AAVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
US-6054457-A Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-25 US disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed